Role of Telomeres in the Development of Cancers

Introductionc-myc, which regulates the expression of the human
          Cancer – although there are overtelomerase reverse transcriptase gene (hTERT) via
hundred types of it, claims millions of lives every yearits promoter region.
throughout the world (American Cancer Society,         The remainder of human cancers
2007); which is a class of diseases in which a groupactivate the Alternative Lengthening of Telomeres
of cells display uncontrolled growth, invade adjacent(ALT) pathway, which relies on
tissues and spread to other locations in the bodyrecombination-mediated elongation and does not need
 and as a result if not treated in time, leads to deathtelomerase. As human telomeres grow shorter,
(Pecorino 2008, p.2). On the other hand, Telomereseventually cells reach the limit of their replicative
are repetitive DNA sequences and protein complexescapacity and progress into senescence. Senescence
added by an enzyme called telomerase and areinvolves the p53 and pRb pathways and leads to the
located at the end of chromosomes, which stabilisesarrest of cell proliferation and plays an important role
the chromosome and protects it from deterioration.in suppression of appearance of cancer (Campisi,
They also have a capping role because telomeres do2005). However, by inactivating the p53 and pRb
not perform homologous recombination and preventpathways further cell proliferation can be achieved;
non homologous end joining; this is because inalso cells entering proliferation after inactivation of
contrast to linear DNA, telomeres are structuresp53 and pRb pathways undergo abnormal
made up of t-loops and four stranded conformationschromosomal rearrangements and leads to genome
named G quadruplexes. In mammalian cells, theinstability, and (almost) all cells die. Rare cells emerge
telomeric sequence is a repetition of a hexanucleotidefrom crisis immortalized through telomere elongation
motif, TTAGGG (Desmaze et al., 2003) varying fromby either activating telomerase or ALT. The first
3 to 20 kilobase pairs in length.description of an ALT cell line demonstrated that the
         Cancer is caused (usually) bytelomeres were highly heterogeneous in length and
abnormalities and/or mutations found in the geneticpredicted a mechanism involving recombination. ALT
material of transformed cells (Pecorino 2008, p.4),cells produce abundant t-circles and if the telomeres
and as time passes, due to the immense damagebecome too short, they will (potentially) unfold from
caused to the cell's defense mechanisms (e.g. DNAtheir presumed closed structure. The cell turns on
repair), these accumulate. When coupled withcertain mechanisms which detects and understands
environmental factors like poor diet, smoking, stressthis uncapping as "DNA damage" and then enters
etc the cells become weaker, quicker; and cancercellular senescence, growth arrest or apoptosis,
probability increases in accordance. There are twodepending on the cell's p53 status. Chromosomal
major types of genes which contribute tofusions can also result in uncapped telomeres. Since
carcinogenesis, called oncogenes and tumorthis damage cannot be repaired in normal somatic
suppressor genes. These genes regulate growth andcells, the cell may even go into apoptosis. Many
division of cells thus mutations within these genes,aging-related diseases are linked to shortened
cause malfunctioning and abnormal growth of cellstelomeres. Organs deteriorate as more and more of
which is the foundation of cancer; so one could saytheir cells die off or enter cellular senescence –
cancer is a genetic disease at the cellular level.eventually leading to the "inevitable".
         Unlike prokaryotes, (most) eukaryotic         Chromosomes that lack telomeres
(this includes humans also) chromosomes are linearremain unstable until they are capped. Broken
which means they have free ends. This detail alonechromosomes that do not gain telomeres can
causes problems due to the fact that DNA replicationundergo sister chromatid fusions involving non
progresses 5' to 3' which leads to discontinuity in thehomologous end joining. These fusions induce
lagging strand, therefore the nucleotide addingchromosome instability resulting from breakage/fusion
enzyme DNA polymerase cannot finish theanaphase bridge (B/F/A) cycles. Coming back to the
polymerisation process neatly when it reaches thedicentric bridge formed at anaphase (mentioned in
end of the chromosomes. A small piece of DNA isintroduction), the two centromeres of a dicentric
left unreplicated at the end of each cell cycle whichchromosome are pulled towards opposite spindle
results in that amount of DNA to be lost and if thispoles creating an anaphase bridge. The chromosome
process carries on the way it does, then this willwould then break, resulting in novel chromosomal
eventually cause the essential, protein-coding regionsrearrangements by fusion of broken ends, and
of the genome to be lost. This is where Telomeresperpetuating a B/F/A cycle. Anaphase bridges can
come into play, since they are at the end ofalso cause whole chromosome losses or the collapse
chromosomes and they only consist of non codingof the cytokinetic process leading to numerical
regions (in the form of repeats); therefore althoughchromosome aberrations. Chromosome
some of it is lost, the cell can divide many timesrearrangements that can theoretically result from
before reaching the essential parts of thesuccessive B/F/A cycles are similar to those
chromosomes. This problem is not present in (most)observed in human carcinomas. This process results in
prokaryotes because the genome is circular and thehighly rearranged chromosomes that eventually
end-problem does not occur because there is noacquire a new telomere through gene amplification
lagging strand.cycles which is a common consequence of genome
         Moving on to humans, it has beeninstability in tumour cells and can be the basis of
observed that somatic cells cease to divide after aoncogene activation and drug resistance.
limited number of divisions, the number ranging from         There is also evidence that
twenty to ninety depending on the age of thechromosomes with shorter telomeres tend to be
person the cell is being taken from; a phenomenonmore affected by radiation; more double strand
known as "cellular aging" (Solomon et al. 2002, p.256);breaks, deletions and translocations seem to occur in
for example, cells taken from a 70 year old man canthese chromosomes (Desmaze et al., 2003). This
divide 20-30 times compared to one extracted fromphenomenon could also increase the chance of
an infant which can divide 80-90 times (Bodnar etcancer progression as this also can also cause
al.,1998). What was observed is that telomeres weregenome instability. All of the above gives strong
much shorter in the older people, and other studiesevidence that telomeres are related with cancer,
(Cancer Research UK, 2010) also show that asdirectly and/or indirectly.
people aged, their risk of being cancer and theConclusion
percentage of people diagnosed with cancer         To conclude, excess shortening of
increased which gave evidence that the two could betelomeres enhances chromosomal instability in cancer
linked to one another. Further research into telomerecells and the loss of one telomere leads to gene
function showed that they had three importantamplification and chromosome imbalances as well as
functions: Prevent DNAses from degrading the endschromosomal instability. Telomeres have important
of the linear DNA molecules, prevent fusion of thefunctions in genome stabilisation; and when they are
ends with other DNA molecules and facilitatenot present or not fully functional there is evidence
replication of the ends of the linear DNA moleculesthat these abnormalities – caused due to the
without loss of essential genetic material (Snustadshortening or total loss of telomeres, help trigger
and Simmons 2006, p.230); and if anything goescancer. Telomeres and cancer are certainly linked but
wrong with these mechanisms it is highly likely thatwhether telomere shortening is the main cause, the
cancer could progress within the cells where theconsequence or is involved in (just) one of the steps
malfunctioning occurs, so the question is: how doesleading to cancer still needs further research.
telomeres play a role in cancer development?         In my opinion, (maybe) in the near
Telomeres and Cancerfuture, measuring telomerase presence/activity could
         Approximately 85% of cancersbe considered a new way to detect cancer; also if
(Pecorino 2008, p.2) occurring in human adults are ofscientists can learn how to stop telomerase
epithelial origin, called carcinomas. These tumoursproduction and/or inhibit its function, they may be
have extremely rearranged karyotypes with a highable to remove cancer by causing cancer cells to age
frequency of translocations which are closely linkedand die. Also further research into why and how
to cancer development due to the generation ofsome cancer cells activate the ALT pathway instead
fusion genes, modification of gene copy number andof telomerase can also give clues in to how cancer
or deregulation of the expression of severalcould be treated and possibly lead to development of
oncogenes. In telomerase knockout mice, telomeredrug treatments. It is easy to say however, as
shortening below a critical length results in increasedscientists discover more secrets about telomeres and
end-to-end chromosome fusions which results intelomerase, their understanding of cancer will increase
dicentric chromosomes and this also generatesin accordance.
instability in the genome. These fused chromosomesReferences
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